Kisspeptin 234

CAS NO.：1145998-81-7
Empirical Formula: C63H78N18O13
Molecular Weight: 1295.41
Update Date: 2026-04-24 14:58:55

What is Kisspeptin 234?

Biological Activity

kisspeptin 234 is a kisspeptin receptor antagonist, with the ability to antagonize kisspeptin-10-induced activation of gpr-54. kisspeptin binds to its cognate receptor (i.e. gpr-54) on neurons that produce gonadotropin-releasing hormone (gnrh), and stimulates their activity, which in turn sends an obligatory signal for gnrh secretion, thereby gating down-stream events supporting reproduction. the development of kisspeptin receptor antagonists may provide a valuable tool for exploring the physiological and pathophysiological roles of kisspeptin in the regulation of reproduction, and could serve as a potential therapeutic agent for treating hormone-dependent disorders of reproduction, such as precocious puberty, endometriosis, as well as metastatic prostate cancer.1. roseweir ak, kauffman as, smith jt, et al. discovery of potent kisspeptin antagonists delineate physiological mechanisms of gonadotropin regulation. journal of neuroscience, 2009, 29(12): 3920-3929.

Storage

Store at -20°C

Properties of Kisspeptin 234

storage temp.	Store at -20°C
solubility	insoluble in DMSO; insoluble in EtOH; ≥4.44 mg/mL in H2O with ultrasonic
form	solid
color	White
Water Solubility	Soluble to 1 mg/ml in water

Safety information for Kisspeptin 234

Computed Descriptors for Kisspeptin 234

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