SETD2-IN-1 TFA
- CAS NO.:2411759-92-5
- Empirical Formula: C24H30F4N4O4
- Molecular Weight: 514.52
- Update Date: 2026-04-22 18:57:36
What is SETD2-IN-1 TFA?
Biological Activity
SETD2-IN-1 TFA is a potent, selective and orally active inhibitor of SETD2 which is a human histone methyltransferase. SETD2-IN-1 TFA has anti-proliferative effects[1].
References
[1]. John Lampe, et al. Substituted indoles and methods of use thereof. WO2020037079A1.
Properties of SETD2-IN-1 TFA
| storage temp. | 4°C, away from moisture |
| solubility | DMSO : 200 mg/mL (388.72 mM; Need ultrasonic) |
| form | Solid |
| color | White to light yellow |
Safety information for SETD2-IN-1 TFA
Computed Descriptors for SETD2-IN-1 TFA
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