L-803,087 Trifluoroacetate
- CAS NO.：217480-26-7
- Empirical Formula: C25H29F2N5O3
- Molecular Weight: 485.53
- MDL number: MFCD09037334
- SAFETY DATA SHEET (SDS)
- Update Date: 2026-09-12 18:55:53
What is L-803,087 Trifluoroacetate?
The Uses of L-803,087 Trifluoroacetate
Somatostatin receptors are often overexpressed in tumours and are potential therapeutic targets. Somatostatin receptor agonists can be used to study signaling pathways related somatostatin receptor. L 803087 is a somatostatin sst4 receptor agonist.
What are the applications of Application
L-803,087 trifluoroacetate is a potent and selective sst4 agonist
Biological Activity
Potent and selective somatostatin sst 4 receptor agonist. K i values are 0.7, 199, 4720, 1280 and 3880 nM for cloned human sst 4 , sst 1 , sst 2 , sst 3 and sst 5 receptors respectively. Facilitates AMPA-mediated hippocampal synaptic responses in vitro and increases kainate-induced seizures in mice in vivo .
Properties of L-803,087 Trifluoroacetate
| Density | 1.33±0.1 g/cm3(Predicted) |
| storage temp. | Store at -20°C |
| solubility | Soluble to 100 mM in DMSO and to 100 mM in ethanol |
| form | Powder |
| pka | 14.54±0.46(Predicted) |
| color | White to light yellow |
Safety information for L-803,087 Trifluoroacetate
Computed Descriptors for L-803,087 Trifluoroacetate
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