KBP-7018
- CAS NO.:1613437-66-3
- Empirical Formula: C31H30N4O5
- Molecular Weight: 538.6
- Update Date: 2026-05-11 19:39:08
What is KBP-7018?
Description
KBP-7018 is a novel, tyrosine kinase-selective inhibitor with potent effects on three fibrotic kinases (c-KIT, PDGFR, and RET). It IC50 values are: c-KIT 10nM; RET 7.6 nM; PDGFR 25nM. KBP-7018 represents a novel multikinase inhibitor with differentiated activity, highly enhanced selectivity, and acceptable PK profiles that will enter phase I clinical trials.
Properties of KBP-7018
| Boiling point: | 812.1±65.0 °C(Predicted) |
| Density | 1.346±0.06 g/cm3(Predicted) |
| pka | 11.05±0.20(Predicted) |
Safety information for KBP-7018
Computed Descriptors for KBP-7018
New Products
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