GW 501516 Sulfone

CAS NO.：1206891-27-1
Empirical Formula: C21H18F3NO5S2
Molecular Weight: 485.5
Update Date: 2026-03-18 11:52:23

What is GW 501516 Sulfone?

The Uses of GW 501516 Sulfone

GW 501516 Sulfone is a urinary metabolite of GW1516 (G931500), a drug candidate potentially enhancing athletic performance. GW 501516 Sulfoxide may be used or doping control purposes.

Definition

ChEBI: GW 501516 sulfone is a sulfone resulting from the oxidation of the sulfur attached to one of the phenyl groups of GW 501516. It is a urinary metabolite of GW 501516 (a failed drug candidate and gene doping agent whose use by athletes has been prohibited by the World Anti-Doping Agency), so detection of the sulfone in sports drugs testing can be used to prove GW 501516 doping. It is a sulfone, a member of 1,3-thiazoles, an aromatic ether, a monocarboxylic acid and an organofluorine compound. It is functionally related to a GW 501516 sulfoxide and a GW 501516.

Properties of GW 501516 Sulfone

Melting point:	>213°C (dec.)
Boiling point:	672.2±65.0 °C(Predicted)
Density	1.423±0.06 g/cm3(Predicted)
storage temp.	Hygroscopic, -20°C Freezer, Under inert atmosphere
solubility	DMSO (Slightly), Methanol (Slightly, Heated)
form	Solid
pka	2.98±0.10(Predicted)
color	White to Off-White
Stability:	Hygroscopic

Safety information for GW 501516 Sulfone

Computed Descriptors for GW 501516 Sulfone

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