GAT-211
- CAS NO.:102704-40-5
- Empirical Formula: C22H18N2O2
- Molecular Weight: 342.39
- MDL number: MFCD02165420
- Update Date: 2026-07-27 17:00:41
What is GAT-211?
Description
GAT211, aslo known as AZ-4, is a small molecule CB1 positive allosteric modulator. GAT211 suppresses allodynia and produces synergistic antiallodynic effects with fatty acid amide hydrolase and monoacylglycerol lipase inhibitors in paclitaxel-treated mice. Positive allosteric modulation of CB1-receptor signaling with GAT211shows promise as a safe and effective analgesic strategy that lacks tolerance, dependence, and abuse liability.
Properties of GAT-211
| storage temp. | Store at -20°C |
| solubility | DMF: 25 mg/ml; DMF:PBS (pH 7.2)(1:3): 0.25 mg/ml; DMSO: 10 mg/ml; Ethanol: 5 mg/ml |
| form | A crystalline solid |
| color | White to off-white |
Safety information for GAT-211
Computed Descriptors for GAT-211
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