GAT-211

CAS NO.：102704-40-5
Empirical Formula: C22H18N2O2
Molecular Weight: 342.39
MDL number: MFCD02165420
Update Date: 2026-04-22 18:57:36

What is GAT-211?

Description

GAT211, aslo known as AZ-4, is a small molecule CB1 positive allosteric modulator. GAT211 suppresses allodynia and produces synergistic antiallodynic effects with fatty acid amide hydrolase and monoacylglycerol lipase inhibitors in paclitaxel-treated mice. Positive allosteric modulation of CB1-receptor signaling with GAT211shows promise as a safe and effective analgesic strategy that lacks tolerance, dependence, and abuse liability.

Properties of GAT-211

storage temp.	Store at -20°C
solubility	DMF: 25 mg/ml; DMF:PBS (pH 7.2)(1:3): 0.25 mg/ml; DMSO: 10 mg/ml; Ethanol: 5 mg/ml
form	A crystalline solid
color	White to off-white

Safety information for GAT-211

Computed Descriptors for GAT-211

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