FR 139317
- CAS NO.：142375-60-8
- Empirical Formula: C33H44N6O5
- Molecular Weight: 604.74
- MDL number: MFCD00467722
- SAFETY DATA SHEET (SDS)
- Update Date: 2026-03-18 11:52:23
What is FR 139317?
The Uses of FR 139317
FR 139317 is a novel, potent endothelin ETA receptor antagonist.
Biological Activity
A highly potent and selective ET A endothelin receptor antagonist (K i values are 1 nM and 7.3 μ M at ET A and ET B subtypes respectively). Active in vivo .
Properties of FR 139317
| Boiling point: | 943.9±65.0 °C(Predicted) |
| Density | 1.27±0.1 g/cm3(Predicted) |
| storage temp. | Desiccate at +4°C |
| solubility | Soluble to 100 mM in 1eq. HCl and to 100 mM in DMSO |
| form | Powder |
| pka | 2.68±0.10(Predicted) |
Safety information for FR 139317
Computed Descriptors for FR 139317
New Products
2,6-Piperidinedione, 3-hydroxy-1-[(4-methoxyphenyl)methyl]- 3-(4-bromo-3-methyl-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)piperidine-2,6-dione 4-Hydroxy-6-methyl-1-(4-methylphenyl)-2-naphthalenecarboxylic acid 2,3-Difluoro-6-methoxybenzyl Chloride KT-474 2-(6-(benzyloxy)-3,4-dihydronaphthalen-2-yl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 3-Oxocyclobutanecarboxylic acid 5-Bromo-2-iodo pyridine Benzofuran-6-carboxylic acid (BFA) 3-Bromo-2-Ethoxy-5-Nitropyridine 3,6-Dichloro-2-Methylpyridine 2-Amino-5-Bromo-3-IodopyridineRelated products of tetrahydrofuran
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