UR-144 N-(5-Hydroxypentyl) β-D-Glucuronide

CAS NO.：1630023-01-6
Empirical Formula: C27H37NO8
Molecular Weight: 503.58458
Update Date: 2023-05-04 17:34:34

What is UR-144 N-(5-Hydroxypentyl) β-D-Glucuronide?

Description

UR-144 is a potent synthetic cannabinoid (CB) which preferentially binds the peripheral CB₂ receptor (K_i = 1.8 nM) over the central CB₁ receptor (K_i = 150 nM). UR-144 N-(5-hydroxypentyl) β-D-glucuronide is an expected major urinary metabolite of UR-144, based on the metabolism of similar cannabimimetics. The physiological and toxicological properties of this compound have not been tested. This product is intended for forensic and research applications.

The Uses of UR-144 N-(5-Hydroxypentyl) β-D-Glucuronide

UR-144 N-(5-Hydroxypentyl) β-D-Glucuronide is the expected major urinary metabolite of UR-144 (P227525), a potent synthetic cannabinoid which has high affinity for the CB2 cannabinoid receptor.

Definition

ChEBI: Beta-d-glucopyranosiduronic acid, 5-[3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1h-indol-1-yl]pentyl is an O-acyl carbohydrate.

Properties of UR-144 N-(5-Hydroxypentyl) β-D-Glucuronide

Boiling point:	709.8±60.0 °C(Predicted)
Density	1.37±0.1 g/cm3(Predicted)
solubility	DMF: 10 mg/ml; DMSO: 5 mg/ml; Ethanol: 12.5 mg/ml; PBS (pH 7.2): 2 mg/ml
form	A crystalline solid
pka	2.83±0.70(Predicted)

Safety information for UR-144 N-(5-Hydroxypentyl) β-D-Glucuronide

Computed Descriptors for UR-144 N-(5-Hydroxypentyl) β-D-Glucuronide

New Products

2-Ethoxyphenol Methyl 2-methoxy-5-sulfamoylbenzoate 3,6-Dichloropyridazine Ethyl 2-chloro-2-(2-(4-methoxyphenyl)hydrazono)acetate 3,6-Dichloro-4-Isopropylpyridazine 2-[(2-Ethoxyphenoxy)methyl]oxirane 4-Morpholinoaniline 2-Chloromethyl-6-methyl-pyridine 1-Indanone tert-Butyl ((1R,2S,5S)-2-amino-5-(dimethylcarbamoyl)cyclohexyl)carbamate 2-Pyridinecarboxaldehdye 6-Methyl-2-pyridinemethanol 4-Bromo-2-fluoro-N-methylbenzamide 3-Azetidinecarboxylic acid N-(2-(4-((4-Fluorobenzyl)carbamoyl)-5-hydroxy-6-methoxypyrimidin-2-yl)propan-2-yl)-5-methyl-1,3,4-oxadiazole-2-carboxamide (R)-4-Boc-morpholine-3-carboxylic acid (Required high chiral purity NLT:99.5%) Tetrahydro-3-(2-methyl-2- nitropropyl)-2H-pyran-2-one 3-Bromo-2-fluorobenzonitrile Desoximetasone Boron Triiodide Nicotinic acid RAPAMYCIN Pentachlorobenzonitrile Budesonide