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HomeProduct name listBKM-120

BKM-120

BKM-120 Structural

What is BKM-120?

The Uses of BKM-120

A selective Class I PI3K inhibitor of p110α, p110β, p110δ and p110γ with IC50s of 50-300 nM.

Definition

ChEBI: An aminopyridine that is 4-(trifluoromethyl)pyridin-2-amine substituted at position 5 by a 2,6-di(morpholin-4-yl)pyrimidin-4-y group. A selective PI3K inhibitor with anti-tumour properties.

Properties of BKM-120

CAS DataBase Reference 1202777-78-3

Safety information for BKM-120

Computed Descriptors for BKM-120

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