BI-4834
- CAS NO.:876371-13-0
- Empirical Formula: C32H47N7O4
- Molecular Weight: 593.76
- Update Date: 2026-01-05 11:31:08
What is BI-4834?
Description
BI-4834 is a potent and selective Polo-like kinase 1 (PLK1) inhibitor. BI-4834 is also analogue (or Me-Too) of BI-2536. In vitro test shows that BI 4834 inhibits PLK1 with IC50=7.6 nm, but with higher selectivity over the related enzyme PLK3 (IC50 198.4 nm) as BI-2536.
Properties of BI-4834
| Density | 1.24±0.1 g/cm3(Predicted) |
| pka | 14.24±0.40(Predicted) |
Safety information for BI-4834
Computed Descriptors for BI-4834
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